Sertaconazole nitrate是一种外用广谱抗真菌药,是用来治疗表面皮肤和粘膜感染的辅助用药.......
Vildagliptin is a dipeptidyl peptidase-4 (CD26) inhibitor. CD26 activates serine......
Y-27632 dihydrochloride is a selective Rho-kinase inhibitor, which suppresses ch......
Pilaralisib (XL147)是一种选择性的可逆I型PI3K抑制剂,作用于PI3Kα/δ/γ,在无细胞试验中IC50为 39 nM/36 nM/23 n......
Nifuroxazide是可渗透细胞的,口服有效的硝基呋喃类止泻药,有效地抑制细胞内STAT1/3/5转录活性的激活,IC50为3 μM。......
Pemetrexed是抗叶酸和抗代谢剂,对TS,DHFR和GARFT的Ki分别为1.3 nM,7.2 nM和65 nM。......
Xylometazoline HCl 是α-adrenoceptor激动剂,常用作鼻血管收缩药,高效作用于α2B肾上腺素受体亚型,EC50为4 μM。......
Telmisartan is an angiotensin II receptor antagonist (ARB) used in the managemen......
Pitavastatin Calcium is a competitive inhibitor of the enzyme HMGCR (HMG-CoA red......
Pazopanib HCl (GW786034 HCl)是一种新型的针对VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Ki......
A77 1726, also known as teriflunomide, is the active metabolite of leflunomide. ......
Sulfasalazine 是一种磺胺剂,是Mesalazine的衍生物,主要用作抗炎剂。......
Sertaconazole nitrate是一种外用广谱抗真菌药,是用来治疗表面皮肤和粘膜感染的辅助用药.......
Semaxanib (SU5416)是VEGFR(Flk-1/KDR)抑制剂,IC50为1.23 μM,比对PDGFRβ的抑制性高20倍,对EGFR,InsR和......
Ruxolitinib (INCB018424)是第一个应用于临床的、有效的、选择性的JAK1/2抑制剂,IC50为3.3 nM/2.8 nM。作用于JAK1,......
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